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Characteristic of approved GLP-1 receptor agonists are listed in Table 1

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Orforglipron is the first small-molecule GLP-1 receptor agonist, taken without food and water restrictions, to successfully complete a Phase 3 trial

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doi: 10.1038/s42255-023-00966-w 62 NovikoffAMullerTD

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doi: 10.1056/NEJMoa1306033

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