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GPCR desensitisation is a real pharmacological risk with any sustained agonist exposure

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Supplementary Validation Method: LCMS/MS For high-sensitivity detection requirements, liquid chromatographytandem mass spectrometry is used for supplementary validation, especially suitable for trace component analysis and metabolic studies

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Es importante subrayar que estos hallazgos son preclnicos: describen fenmenos observados en sistemas controlados de laboratorio y no constituyen evidencia de eficacia o seguridad en humanos

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*** Ephedrine and methylephedrine: Prohibited when the concentration of either in urine is greater than 10 micrograms per millilitre

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